SCHEMBL25810490

SCHEMBL25810490

COC(=O)C(C)c1cccc(C(N)=O)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.70
PTGS2 P35354 4/20 0.70
PARP1 P09874 8/20 0.51
MAPT P10636 2/20 0.47
CXCR1 P25024 2/20 0.47
CXCR2 P25025 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HPGD P15428 2/20 0.47
RECQL P46063 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPK1 P28482 1/20 0.47
PMP22 Q01453 1/20 0.47
SLC22A6 Q4U2R8 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CXCL8 P10145 1/20 0.47
THPO P40225 1/20 0.47
HIF1A Q16665 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8376478 0.89 PTGS1 (0.55) PTGS1PTGS2PARP1MAPTCXCR1
SCHEMBL31477369 0.85 PTGS1 (0.72) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL9030430 0.85 PTGS1 (0.72) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL31455828 0.85 PTGS1 (0.77) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL8754918 0.83 PTGS1 (1.00) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL577323 0.83 PTGS1 (1.00) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL12935378 0.83 PTGS1 (1.00) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL9086931 0.83 PTGS1 (1.00) PTGS1PTGS2MAPTCXCR1CXCR2
SCHEMBL14661109 0.83 PARP1 (0.50) PTGS1PTGS2PARP1SMN1; SMN2PARP10
SCHEMBL11132637 0.81 PTGS1 (0.70) PTGS1PTGS2PARP1MAPTCXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230219961-A1 Pyridine acetamide derivative serving as CDK inhibitor, and preparation method therefor and use thereof Suzhou Alphama Biotechnology Co., Ltd. (CN) 2023-07-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219961-A1 Pyridine acetamide derivative serving as CDK inhibitor, and preparation method therefor and use thereof CDK9, CDK7, CDK8 PTGS1 1205/4885PTGS2 2365/4885PARP1 828/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.