SCHEMBL25815883

SCHEMBL25815883

O=C(CS)NC1CCN(CCc2ccccc2)CC1

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.80
DRD4 P21917 4/20 0.63
CXCR3 P49682 2/20 0.61
HTR2A P28223 1/20 0.56
ACHE P22303 1/20 0.52
POLB P06746 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5504017 0.88 SIGMAR1 (0.82) SIGMAR1DRD4CXCR3HTR2AACHE
SCHEMBL10648926 0.86 SIGMAR1 (0.80) SIGMAR1DRD4CXCR3HTR2AACHE
SCHEMBL27430491 0.86 SIGMAR1 (0.79) SIGMAR1DRD4CXCR3HTR2AACHE
Oxalic Acid SCHEMBL17512169 0.84 SIGMAR1 (0.76) SIGMAR1DRD4CXCR3HTR2AACHE
Oxalic Acid SCHEMBL21836756 0.84 SIGMAR1 (0.76) SIGMAR1DRD4CXCR3HTR2AACHE
SCHEMBL8023030 0.83 SIGMAR1 (0.75) SIGMAR1DRD4CXCR3HTR2AACHE
SCHEMBL17512174 0.82 DRD4 (0.76) SIGMAR1DRD4HTR2A
SCHEMBL31486979 0.81 SIGMAR1 (0.71) SIGMAR1DRD4
SCHEMBL17512172 0.80 SIGMAR1 (0.70) SIGMAR1DRD4CXCR3HTR2A
SCHEMBL10514979 0.80 SIGMAR1 (0.79) SIGMAR1DRD4CXCR3HTR2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023133135-A2 SMALL MOLECULE ADRENORECEPTOR ANTAGONISTS AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2023-07-13 WO disclosed