SCHEMBL2581908

SCHEMBL2581908

CC(N)c1nc2cccc(S(C)(=O)=O)c2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
ALOX12 P18054 1/20 0.37
TAAR1 Q96RJ0 1/20 0.35
TYK2 P29597 4/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
CDC7 O00311 1/20 0.32
PIM1 P11309 1/20 0.32
CSNK2B P67870 1/20 0.32
CSNK2A1 P68400 1/20 0.32
MPO P05164 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
HDAC11 Q96DB2 1/20 0.30
DRD4 P21917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2509772 1.00 PARP1 (0.42) PARP1ALOX12TAAR1TYK2NPC1
SCHEMBL12221753 0.76 PARP1 (0.40) PARP1TAAR1KMT2A
SCHEMBL2509581 0.75 PARP1 (0.39) PARP1TAAR1NPC1RAB9A
SCHEMBL8034264 0.75 NPC1 (0.34) ALOX12TYK2NPC1RAB9AKMT2A
SCHEMBL12263337 0.74 PIK3CG (0.44)
SCHEMBL5859162 0.72 KDM4E (0.39) NPC1RAB9AKMT2ADRD4
SCHEMBL2504431 0.71 PIK3CD (0.53)
SCHEMBL524001 0.67 TAAR1 (0.68) PARP1ALOX12TAAR1NPC1RAB9A
SCHEMBL12737571 0.67 TAAR1 (0.68) PARP1ALOX12TAAR1NPC1RAB9A
SCHEMBL8330903 0.67 TAAR1 (0.68) PARP1ALOX12TAAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552908-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES Amgen Inc. (US) 2013-02-06 EP disclosed
WO-2011123751-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2011-10-06 WO disclosed