SCHEMBL2582335

SCHEMBL2582335

Cc1ccc(CNC(=O)c2noc3c2CN(C(=S)Nc2c(F)c(F)c(F)c(F)c2F)CC3)o1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.45
ALDH1A1 P00352 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.40
LMNA P02545 4/20 0.39
HPGD P15428 2/20 0.39
KMT2A Q03164 3/20 0.39
TSHR P16473 3/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPT P10636 1/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
ATM Q13315 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2586908 0.79 ALDH1A1 (0.58) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL2580456 0.78 HSP90AA1 (0.44) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL4270038 0.77 NPC1 (0.38) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL2585248 0.73 POLB (0.46) HSP90AA1ALDH1A1SMN1; SMN2LMNAKMT2A
SCHEMBL15300340 0.69 CHRM3 (0.33) HSP90AA1HPGDKMT2AMEN1RAB9A
SCHEMBL2582213 0.69 GAA (0.57) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL2587252 0.67 ALDH1A1 (0.57) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL4268590 0.66 MAPT (0.58) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL2580833 0.65 ALDH1A1 (0.53) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL2586734 0.64 HSP90AA1 (0.55) HSP90AA1ALDH1A1SMN1; SMN2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed