SCHEMBL25824383

SCHEMBL25824383

N=C/C(=C\N)c1ccc2nc(Nc3ccc(C4CCOCC4)cc3)c3nccn3c2c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 14/20 0.43
SYK P43405 1/20 0.43
IRAK4 Q9NWZ3 2/20 0.40
LCK P06239 1/20 0.37
JAK3 P52333 1/20 0.37
MAST3 O60307 4/20 0.36
MAPKAPK5 Q8IW41 1/20 0.36
IKBKB O14920 1/20 0.35
MAPK9 P45984 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25822757 0.81 SYK (0.47) MAPK8SYKLCKJAK3MAPKAPK5
SCHEMBL26184439 0.79 MAPK8 (0.38) MAPK8SYKMAST3MAPKAPK5IKBKB
SCHEMBL25823859 0.79 MAPK8 (0.40) MAPK8SYKMAST3MAPKAPK5
SCHEMBL25823409 0.78 MAPKAPK5 (0.43) MAPK8SYKLCKMAPKAPK5IKBKB
SCHEMBL25822697 0.75 SYK (0.53) MAPK8SYKLCKMAPKAPK5
SCHEMBL25823831 0.73 SYK (0.49) SYK
SCHEMBL21949418 0.68 IRAK4 (0.43) IRAK4
SCHEMBL21949415 0.68 PYGM (0.43) IRAK4
SCHEMBL15552071 0.67 SYK (0.60) SYKLCKJAK3
SCHEMBL25822712 0.66 MAPT (0.58) SYKMAPKAPK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230219960-A1 1H-PYRAZOLE DERIVATIVE AND APPLICATION THEREOF AS DUAL TARGET INHIBITOR OF SYK AND VEGFR2 OCUMENSION THERAPEUTICS (SUZHOU) CO., LTD. (CN) 2023-07-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219960-A1 1H-PYRAZOLE DERIVATIVE AND APPLICATION THEREOF AS DUAL TARGET INHIBITOR OF SYK AND VEGFR2 SYK, KDR, FLT1 MAPK8 637/4885SYK 1/4885IRAK4 106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.