SCHEMBL25833569

SCHEMBL25833569

O=C(Nc1nc2ccc(-c3ccc(C(F)(F)F)cc3)cc2s1)[C@@H]1C2C=CC(C2)[C@@H]1C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.62
CYP2D6 P10635 1/20 0.56
ABL1 P00519 9/20 0.55
DYRK1A Q13627 1/20 0.50
ITK Q08881 1/20 0.50
CSNK1D P48730 3/20 0.48
PIK3CG P48736 1/20 0.47
PIK3CD O00329 1/20 0.46
ACP1 P24666 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25262799 1.00 ALDH1A1 (0.62) ALDH1A1CYP2D6ABL1DYRK1AITK
SCHEMBL30450160 1.00 ALDH1A1 (0.62) ALDH1A1CYP2D6ABL1DYRK1AITK
SCHEMBL30451396 0.92 ALDH1A1 (0.67) ALDH1A1CYP2D6DYRK1ACSNK1DACP1
SCHEMBL25300056 0.92 ALDH1A1 (0.67) ALDH1A1CYP2D6DYRK1ACSNK1DACP1
SCHEMBL25833329 0.92 ALDH1A1 (0.67) ALDH1A1CYP2D6DYRK1ACSNK1DACP1
SCHEMBL30450144 0.92 ALDH1A1 (0.59) ALDH1A1CYP2D6ABL1DYRK1AITK
SCHEMBL25833539 0.92 ALDH1A1 (0.59) ALDH1A1CYP2D6ABL1DYRK1AITK
SCHEMBL25299562 0.92 ALDH1A1 (0.59) ALDH1A1CYP2D6ABL1DYRK1AITK
SCHEMBL25306737 0.89 ALDH1A1 (0.66) ALDH1A1ABL1ITKPIK3CG
SCHEMBL30450121 0.89 ALDH1A1 (0.66) ALDH1A1ABL1ITKPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131649-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-07-13 WO disclosed