SCHEMBL25834339

SCHEMBL25834339

O=C(Nc1nc2ccc(Nc3ccc(OC(F)(F)F)cn3)cc2s1)[C@@H]1C2C=CC(C2)[C@@H]1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
DYRK1A Q13627 1/20 0.46
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
ACP1 P24666 1/20 0.41
POLB P06746 1/20 0.41
CASP6 P55212 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CSNK1D P48730 5/20 0.40
ITK Q08881 2/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30450317 1.00 ALDH1A1 (0.53) ALDH1A1DYRK1AHDAC3HDAC4HDAC1
SCHEMBL25259129 1.00 ALDH1A1 (0.53) ALDH1A1DYRK1AHDAC3HDAC4HDAC1
SCHEMBL30450379 0.88 ALDH1A1 (0.55) ALDH1A1DYRK1AACP1POLBCSNK1D
SCHEMBL25307365 0.88 ALDH1A1 (0.55) ALDH1A1DYRK1AACP1POLBCSNK1D
SCHEMBL30451400 0.87 ALDH1A1 (0.58) ALDH1A1DYRK1APOLBCASP6TDP1
SCHEMBL25299150 0.87 ALDH1A1 (0.58) ALDH1A1DYRK1APOLBCASP6TDP1
SCHEMBL25834103 0.87 ALDH1A1 (0.58) ALDH1A1DYRK1APOLBCASP6TDP1
SCHEMBL25304740 0.86 ALDH1A1 (0.63) ALDH1A1DYRK1AHDAC3HDAC4HDAC1
SCHEMBL30450222 0.84 ALDH1A1 (0.60) ALDH1A1DYRK1AHDAC3HDAC4HDAC1
SCHEMBL25304574 0.84 ALDH1A1 (0.60) ALDH1A1DYRK1AHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131649-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-07-13 WO disclosed