SCHEMBL25834913

SCHEMBL25834913

CNC(=O)c1ncccc1Nc1nc(Nc2ccc3c(c2)CC[C@@H](N2CCCC2)CC3)ncc1Cl

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MET P08581 12/20 0.56
INSR P06213 2/20 0.56
SLC2A1 P11166 2/20 0.56
ALK Q9UM73 10/20 0.53
EGFR P00533 3/20 0.51
PTK2 Q05397 1/20 0.49
MAP4K1 Q92918 1/20 0.49
MAPK8 P45983 1/20 0.49
MAPK9 P45984 1/20 0.49
MAPK10 P53779 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24073380 1.00 MET (0.56) METINSRSLC2A1ALKEGFR
SCHEMBL24073480 0.90 MET (0.69) METINSRSLC2A1ALKEGFR
SCHEMBL24073717 0.90 MET (0.69) METINSRSLC2A1ALKEGFR
SCHEMBL25834891 0.89 MET (0.56) METINSRALKEGFRPTK2
SCHEMBL24073743 0.89 MET (0.56) METINSRALKEGFRPTK2
SCHEMBL24073388 0.89 MET (0.58) METINSRSLC2A1ALK
SCHEMBL30266404 0.88 MET (0.58) METINSRSLC2A1ALKEGFR
SCHEMBL25834885 0.88 MET (0.58) METINSRSLC2A1ALKEGFR
SCHEMBL24073724 0.88 MET (0.58) METINSRSLC2A1ALKEGFR
SCHEMBL24073769 0.87 MET (0.52) METINSRALKEGFRMAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230227484-A1 PYRIMIDINE COMPOUND AS AXL INHIBITOR NANJING CHIA TAI TIANQING PHARMACEUTICAL CO., LTD. (CN) 2023-07-20 US disclosed
US-20230227484-A1 PYRIMIDINE COMPOUND AS AXL INHIBITOR NANJING CHIA TAI TIANQING PHARMACEUTICAL CO., LTD. (CN) 2023-07-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227484-A1 PYRIMIDINE COMPOUND AS AXL INHIBITOR AXL, FLT3, TYMP MET 356/4885INSR 1450/4885SLC2A1 4568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.