SCHEMBL25837880

SCHEMBL25837880

CC(C)c1cc2c(c([C@@H]3CCCN3)c1)CN(C(=O)C(C(F)(F)F)C(F)(F)F)CC2

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.34
CFTR P13569 1/20 0.31
DPP4 P27487 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25837751 0.85 PDK2 (0.38) MAPK1
SCHEMBL25837884 0.83 MAPK1 (0.33) MAPK1DPP4DPP7
SCHEMBL25838478 0.82
SCHEMBL25837881 0.82 MAPK1 (0.33) MAPK1DPP4DPP7
SCHEMBL25837971 0.79 CHRNB2 (0.36) MAPK1HTR2AHTR2C
SCHEMBL25838477 0.79 PRMT5 (0.31)
SCHEMBL25838492 0.79 PRMT5 (0.30)
SCHEMBL25837876 0.78 PDK2 (0.37)
SCHEMBL25838332 0.77 GLRA1 (0.38)
SCHEMBL25838323 0.77 GFER (0.45) MAPK1CFTRHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed