SCHEMBL25838498

SCHEMBL25838498

CCc1cc2c(c([C@@H]3CCCN3)c1)CN(C(=O)C(C)(C)O)CC2

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
PRMT5 O14744 3/20 0.33
WDR77 Q9BQA1 3/20 0.33
RIPK1 Q13546 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
F2 P00734 1/20 0.30
MMP8 P22894 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25837739 0.85 DPP4 (0.31) DPP4DPP7PRMT5WDR77
SCHEMBL25837977 0.79 NAMPT (0.33) PRMT5WDR77RIPK1CYP2D6CYP1A2
SCHEMBL25837751 0.78 PDK2 (0.38)
SCHEMBL25303363 0.75 MAP3K12 (0.39)
SCHEMBL30068777 0.75 MAP3K12 (0.39)
SCHEMBL25303364 0.75 MAP3K12 (0.39)
SCHEMBL25837984 0.75 MAPT (0.35) HPGDHTTHDAC6
SCHEMBL25837884 0.74 MAPK1 (0.33) DPP4DPP7ESR1ESR2
SCHEMBL25302601 0.74 PAK1 (0.40)
SCHEMBL25302603 0.74 PAK1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed