SCHEMBL25839031

SCHEMBL25839031

Cc1cnc2[nH]cc(-c3nc(C(=O)N(C)C)co3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.42
JAK3 P52333 2/20 0.42
ABL1 P00519 3/20 0.38
JAK1 P23458 1/20 0.38
MAP4K1 Q92918 6/20 0.37
MAP3K11 Q16584 1/20 0.36
CYP3A4 P08684 4/20 0.36
CAMKK2 Q96RR4 1/20 0.36
IGF1R P08069 3/20 0.35
HSD17B1 P14061 1/20 0.35
CLK1 P49759 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK2 Q92630 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
TNIK Q9UKE5 1/20 0.34
RIPK1 Q13546 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21592657 0.78 MAP4K1 (0.50) JAK2JAK3ABL1MAP4K1MAP3K11
SCHEMBL25838965 0.78 MAP3K11 (0.52) ABL1MAP4K1MAP3K11CYP3A4CAMKK2
SCHEMBL21592549 0.76 MAP4K1 (0.53) JAK2JAK3MAP4K1MAP3K11CAMKK2
SCHEMBL28769136 0.76 MAP4K1 (0.54) JAK2JAK3ABL1MAP4K1MAP3K11
SCHEMBL31553234 0.76 MAP4K1 (0.54) JAK2JAK3ABL1MAP4K1MAP3K11
SCHEMBL21592847 0.73 MAP4K1 (0.61) JAK2JAK3MAP4K1MAP3K11CAMKK2
SCHEMBL21592554 0.73 MAP4K1 (0.53) ABL1MAP4K1MAP3K11CAMKK2DYRK1A
SCHEMBL28502410 0.73 JAK2 (0.44) JAK2JAK3JAK1CYP3A4CAMKK2
SCHEMBL30267564 0.67 AXL (0.50) CYP3A4CAMKK2
SCHEMBL13941746 0.67 AXL (0.50) CYP3A4CAMKK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed