SCHEMBL25839040

SCHEMBL25839040

Cc1cnc2[nH]cc(C(=O)c3ccccc3Cl)c2c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 8/20 0.60
PKN1 Q16512 1/20 0.56
PAK4 O96013 1/20 0.53
BTK Q06187 6/20 0.47
AXL P30530 1/20 0.46
BRAF P15056 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.45
AAK1 Q2M2I8 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3705469 0.78 CYP3A4 (0.52) PAK1AXLBRAFCYP3A4CYP2C19
SCHEMBL3705466 0.78 CYP3A4 (0.52) PAK1BTKAXLBRAFCYP3A4
SCHEMBL13941746 0.77 AXL (0.50) AXLBRAFCYP3A4CYP2C19AAK1
SCHEMBL30267564 0.77 AXL (0.50) AXLBRAFCYP3A4CYP2C19AAK1
SCHEMBL4570625 0.77 BRAF (0.56) PAK1AXLBRAFCYP3A4CYP2C19
SCHEMBL12146867 0.76 CYP2C19 (0.47) AXLBRAFCYP3A4CYP2C19AAK1
SCHEMBL25251383 0.75 LMNA (0.56) AXLBRAFCYP3A4CYP2C19KMT2A
SCHEMBL30566010 0.75 LMNA (0.56) AXLBRAFCYP3A4CYP2C19KMT2A
SCHEMBL857306 0.75 PAK1 (0.48) PAK1PKN1PAK4BTKAXL
SCHEMBL3710853 0.75 NEK2 (0.50) PAK1PAK4AXLBRAFCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed