SCHEMBL25839042

SCHEMBL25839042

Cc1cnc2[nH]cc(C(O)c3ccccc3Cl)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
BRD4 O60885 1/20 0.39
JAK2 O60674 1/20 0.37
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
AXL P30530 2/20 0.36
CDK8 P49336 1/20 0.36
TNIK Q9UKE5 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25839041 0.86 HDAC3 (0.40) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL12140718 0.83 BRD4 (0.43) BRD4JAK2AXLCDK8TNIK
SCHEMBL16060878 0.80 BRD4 (0.64) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL21873016 0.80 CYP3A4 (0.38) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL12140726 0.73 AXL (0.39) JAK2AXLCDK8TNIKITK
SCHEMBL12140733 0.73 AXL (0.39) JAK2AXLCDK8TNIKITK
SCHEMBL12140715 0.73 AXL (0.39) JAK2AXLCDK8TNIKITK
SCHEMBL17998678 0.73 PRMT5 (0.43) CAMKK2
SCHEMBL91445 0.72 AXL (0.41) JAK2AXLBTKITK
SCHEMBL1358648 0.72 ITK (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed