SCHEMBL25839041

SCHEMBL25839041

Cc1cnc2[nH]cc(C(C)c3ccccc3Cl)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
JAK2 O60674 2/20 0.38
AXL P30530 2/20 0.37
CDK8 P49336 1/20 0.37
TNIK Q9UKE5 1/20 0.37
GSK3B P49841 1/20 0.36
CAMKK2 Q96RR4 1/20 0.35
ITK Q08881 2/20 0.35
PLK4 O00444 1/20 0.35
AURKA O14965 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25839042 0.86 HDAC3 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL12140726 0.82 AXL (0.39) JAK2AXLCDK8TNIKGSK3B
SCHEMBL12140733 0.82 AXL (0.39) JAK2AXLCDK8TNIKGSK3B
SCHEMBL12140715 0.82 AXL (0.39) JAK2AXLCDK8TNIKGSK3B
SCHEMBL17998678 0.77 PRMT5 (0.43) CAMKK2CYP3A4CYP2C19CYP2C9PRMT5
SCHEMBL1357489 0.75 ITK (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL91445 0.73 AXL (0.41) JAK2AXLITKCYP3A4CYP2C19
SCHEMBL12140718 0.73 BRD4 (0.43) JAK2AXLCDK8TNIKGSK3B
SCHEMBL25839040 0.70 PAK1 (0.60) AXLCYP3A4CYP2C19PAK1BTK
SCHEMBL24067233 0.70 CYP2C9 (0.37) CYP3A4CYP2C19CYP2C9PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed