SCHEMBL25839062

SCHEMBL25839062

CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc3c(c2)CCNC3)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AXL P30530 5/20 0.53
NEK2 P51955 1/20 0.46
ALK Q9UM73 10/20 0.45
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
MAP4K1 Q92918 3/20 0.42
BPTF Q12830 1/20 0.42
INSR P06213 4/20 0.41
BTK Q06187 1/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25839009 0.86 AXL (0.71) AXLNEK2ALKAURKAAURKB
SCHEMBL885317 0.71 AXL (0.73) AXLNEK2ALKAURKAAURKB
SCHEMBL24072923 0.68 AXL (0.76) AXLNEK2ALKAURKAAURKB
SCHEMBL24073783 0.68 AXL (0.76) AXLNEK2ALKAURKAAURKB
SCHEMBL19831512 0.68 ALK (0.65) AXLALKINSRMET
SCHEMBL886555 0.67 AXL (0.77) AXLNEK2ALKAURKAAURKB
SCHEMBL23533823 0.67 MAP4K1 (0.72) ALKMAP4K1MET
SCHEMBL31173541 0.67 AXL (0.76) AXLNEK2ALKAURKAAURKB
SCHEMBL25837783 0.67 AXL (0.76) AXLNEK2ALKAURKAAURKB
SCHEMBL886365 0.67 AXL (0.76) AXLNEK2ALKAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134582-A1 PYRIMIDINE-2,4-DIAMINE DERIVATIVES AS WELL AS PREPARATION METHOD THEREFOR AND USE THEREOF 上海立森印迹医药技术有限公司 2023-07-20 WO disclosed