SCHEMBL25839063

SCHEMBL25839063

Cc1cnc2[nH]cc(-c3cccnc3)c2c1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 12/20 0.63
PIK3CA P42336 2/20 0.63
NTRK1 P04629 1/20 0.63
NEK1 Q96PY6 2/20 0.60
KIT P10721 1/20 0.58
DYRK1B Q9Y463 1/20 0.58
CLK1 P49759 7/20 0.57
MAPK1 P28482 1/20 0.55
CCNT1 O60563 1/20 0.53
CCNA2 P20248 1/20 0.53
CDK2 P24941 1/20 0.53
CDK9 P50750 1/20 0.53
PLCG1 P19174 1/20 0.53
AXL P30530 1/20 0.52
CDK8 P49336 1/20 0.52
TNIK Q9UKE5 1/20 0.52
GSK3B P49841 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20319074 0.87 DYRK1A (0.58) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL25785930 0.85 AXL (0.71) DYRK1ANTRK1NEK1CDK2AXL
SCHEMBL26174749 0.84 NEK1 (0.48) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL20319120 0.84 DYRK1A (0.66) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL17952128 0.84 NTRK1 (0.62) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL19068218 0.83 DYRK1A (0.64) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL17951904 0.83 DYRK1A (0.74) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL15333224 0.83 DYRK1A (0.74) DYRK1APIK3CANTRK1NEK1KIT
SCHEMBL25839064 0.82 DYRK1A (0.56) DYRK1ANTRK1KITDYRK1BCLK1
SCHEMBL856823 0.82 CDC7 (0.68) DYRK1APIK3CANTRK1NEK1DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed