SCHEMBL25839481

SCHEMBL25839481

CNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(C(=O)OC)cc2)ncc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 8/20 0.68
PTK2 Q05397 6/20 0.68
INSR P06213 3/20 0.68
AURKA O14965 2/20 0.68
MET P08581 2/20 0.68
MAPK9 P45984 2/20 0.68
MAPK10 P53779 2/20 0.68
CDC7 O00311 1/20 0.68
PLK4 O00444 1/20 0.68
CHEK1 O14757 1/20 0.68
DCLK1 O15075 1/20 0.68
MAPK13 O15264 1/20 0.68
PDPK1 O15530 1/20 0.68
DYRK3 O43781 1/20 0.68
JAK2 O60674 1/20 0.68
ROCK2 O75116 1/20 0.68
RPS6KA5 O75582 1/20 0.68
PRKD3 O94806 1/20 0.68
MAP4K4 O95819 1/20 0.68
PAK4 O96013 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25299781 0.84 PTK2 (0.65) ALKPTK2INSRAURKAMET
SCHEMBL25304543 0.83 PTK2 (0.66) ALKPTK2INSRAURKAMET
SCHEMBL19601638 0.82 ALK (0.65) ALKPTK2INSRAURKAMET
SCHEMBL12570609 0.81 ALK (0.67) ALKPTK2INSRAURKAMET
SCHEMBL12893063 0.81 ALK (0.77) ALKPTK2INSRAURKAMET
SCHEMBL2592094 0.78 ALK (0.67) ALKPTK2INSRAURKAMET
SCHEMBL10207667 0.78 ALK (0.67) ALKPTK2INSRAURKAMET
SCHEMBL2595611 0.78 EGFR (0.65) ALKPTK2INSRAURKAMET
SCHEMBL28384265 0.78 ALK (0.76) ALKPTK2INSRAURKAMET
SCHEMBL21437921 0.78 AXL (0.70) ALKPTK2AURKAMAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134582-A1 PYRIMIDINE-2,4-DIAMINE DERIVATIVES AS WELL AS PREPARATION METHOD THEREFOR AND USE THEREOF 上海立森印迹医药技术有限公司 2023-07-20 WO disclosed
CN-116444488-A Pyrimidine-2, 4-diamine derivative and preparation method and application thereof 上海立森印迹医药技术有限公司 2023-07-18 CN disclosed