SCHEMBL25856422

SCHEMBL25856422

C#Cc1ccc(-c2nnc(N)nc2C)c(O)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.36
ADORA1 P30542 7/20 0.36
ALDH1A1 P00352 3/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 2/20 0.33
ATM Q13315 1/20 0.33
MAPT P10636 3/20 0.33
TSHR P16473 3/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ADORA2B P29275 2/20 0.33
HTT P42858 2/20 0.32
NLRP3 Q96P20 3/20 0.31
MAPK1 P28482 2/20 0.31
CDC7 O00311 1/20 0.31
CDK2 P24941 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24696097 0.86 NLRP3 (0.42) ADORA2AADORA1ALDH1A1LMNAKDM4E
SCHEMBL25861616 0.81 NLRP3 (0.39) NLRP3
SCHEMBL25859022 0.79 EGLN1 (0.37) NLRP3
SCHEMBL25856432 0.78 NLRP3 (0.38) NLRP3
SCHEMBL24695713 0.78 ADORA2A (0.46) ADORA2AADORA1ALDH1A1LMNAKDM4E
SCHEMBL24695931 0.78 ADORA2A (0.46) ADORA2AADORA1ALDH1A1LMNAKDM4E
SCHEMBL31314292 0.77 NLRP3 (0.30) KMT2AATMNLRP3
SCHEMBL31314251 0.76 CACNA2D1 (0.33) KMT2AATMTSHR
SCHEMBL31495957 0.75 NLRP3 (0.34) NLRP3
SCHEMBL24695420 0.74 NLRP3 (0.53) ADORA2AADORA1KDM4ENLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed