SCHEMBL25857097

SCHEMBL25857097

Cc1ccc(CCN(C)C)cc1Br

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 7/20 0.57
HRH3 Q9Y5N1 6/20 0.50
HTR7 P34969 4/20 0.49
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
HTR2A P28223 2/20 0.39
HTR1A P08908 2/20 0.38
CHRNA7 P36544 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR1E P28566 1/20 0.38
HTR2B P41595 1/20 0.38
HTR5A P47898 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8507804 0.82 HRH3 (0.56) TAAR1HRH3HTR7MEN1ALDH1A1
SCHEMBL25430010 0.79 TAAR1 (0.55) TAAR1HRH3HTR7MEN1ALDH1A1
SCHEMBL20918900 0.78 SKP2 (0.46) MEN1ALDH1A1MAPTKMT2A
SCHEMBL9378588 0.77 HPGD (0.40) HRH3MEN1ALDH1A1MAPTKMT2A
SCHEMBL27798768 0.77 SKP2 (0.59) TAAR1HRH3HTR7MEN1ALDH1A1
SCHEMBL6915886 0.76 TAAR1 (0.50) TAAR1HTR7ALDH1A1TP53CYP1A2
SCHEMBL1099654 0.76 ALDH1A1 (0.47) MEN1ALDH1A1CYP1A2MAPTCYP2C19
SCHEMBL17704659 0.74 ESR1 (0.48) MEN1ALDH1A1MAPTCYP2C19KMT2A
SCHEMBL3931779 0.74 SKP2 (0.61) MEN1ALDH1A1TP53CYP1A2MAPT
SCHEMBL18762839 0.73 HRH3 (0.84) TAAR1HRH3MEN1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4212531-A1 AZAINDOLE DERIVATIVES AND THEIR USE AS ERK KINASE INHIBITORS AGV Discovery (FR) 2023-07-19 EP disclosed