SCHEMBL2585775

SCHEMBL2585775

Cc1cnc2[nH]cc(Cc3cnc(Nc4ccccc4C(C)(C)C)nc3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.56
CYP2C9 P11712 10/20 0.56
CYP2C19 P33261 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2579682 0.82 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19
SCHEMBL2537798 0.81 CYP3A4 (0.55) CYP3A4CYP2C9CYP2C19
Ammonia Solution, Strong SCHEMBL2546398 0.80 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19
SCHEMBL2540422 0.77 CYP2C9 (0.53) CYP3A4CYP2C9CYP2C19
SCHEMBL2537090 0.76 CYP2C9 (0.60) CYP3A4CYP2C9CYP2C19
SCHEMBL2540030 0.76 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19
SCHEMBL19366349 0.76 CYP3A4 (0.57) CYP3A4CYP2C9CYP2C19
SCHEMBL2542238 0.74 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19
SCHEMBL1883624 0.74 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19
SCHEMBL2537966 0.74 CYP2C9 (0.63) CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560972-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR Plexxikon, Inc. (US) 2013-02-27 EP disclosed
WO-2011133637-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON, INC. (US) 2011-10-27 WO disclosed