SCHEMBL25858580

SCHEMBL25858580

COC(=O)c1cnn(CCN2CC(N)(N)C2)n1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33
KMT2A Q03164 2/20 0.32
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAPK1 P28482 1/20 0.31
PDE1C Q14123 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23991233 0.87 DPP4 (0.33) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL5656055 0.77 KCNA5 (0.38) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL31729267 0.76 KCNA5 (0.38) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL23989812 0.76 KCNA5 (0.38) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL20139438 0.75 KCNA5 (0.37) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL24768373 0.74
SCHEMBL1412434 0.74 MAPK1 (0.40) KCNA5KMT2AMEN1NPC1RAB9A
SCHEMBL23991141 0.73 KCNA5 (0.36) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL20139419 0.73 KCNA5 (0.33) KCNA5KMT2APOLBTDP1MEN1
SCHEMBL23985960 0.72 ALDH1A1 (0.36) KCNA5KMT2APOLBTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11702422-B2 Imidazopyridazines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-07-18 US disclosed
US-11702422-B2 Imidazopyridazines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-07-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11702422-B2 Imidazopyridazines as modulators of IL-17 IL17A, IL23R, IL15 KCNA5 2932/4885AKT1 3322/4885AKT2 2966/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.