SCHEMBL25859374

SCHEMBL25859374

CC(C)(C)OC(=O)NCNc1ccccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.50
MALT1 Q9UDY8 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
KDM4A O75164 1/20 0.42
BCHE P06276 1/20 0.41
IDO1 P14902 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
SYK P43405 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
HDAC3 O15379 2/20 0.39
HDAC2 Q92769 2/20 0.39
NCOR2 Q9Y618 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2975056 0.87 MALT1 (0.54) HDAC1MALT1LMNAPOLBKDM4A
SCHEMBL29655427 0.87 MALT1 (0.54) HDAC1MALT1LMNAPOLBKDM4A
SCHEMBL23736432 0.85 MALT1 (0.43) HDAC1MALT1LMNAPOLBKDM4A
SCHEMBL4565908 0.85 HDAC1 (0.50) HDAC1MALT1LMNAPOLBKDM4A
SCHEMBL22605515 0.85 BRD4 (0.49) HDAC1MALT1BCHECA12CA1
SCHEMBL22121240 0.83 HDAC1 (0.49) HDAC1MALT1LMNAPOLBKDM4A
SCHEMBL23997305 0.83 HDAC1 (0.63) HDAC1KDM4ACA12CA1CA7
SCHEMBL30336954 0.83 HDAC1 (0.63) HDAC1KDM4ACA12CA1CA7
SCHEMBL28514702 0.82 IDO1 (0.47) HDAC1MALT1LMNABCHEIDO1
SCHEMBL21071330 0.81 ADORA2A (0.47) HDAC1MALT1LMNAPOLBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023136942-A1 SYNTHETIC INTERMEDIATES AND IMPROVED PROCESSES FOR PREPARING ROCK INHIBITORS AERIE PHARMACEUTICALS, INC. (US) 2023-07-20 WO disclosed