SCHEMBL25864424

SCHEMBL25864424

COC1(C)CC(Nc2nnc(-c3ccc(/C=C/C4CC4)cc3O)c3c2CCCC3)C1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 6/20 0.53
IL1B P01584 6/20 0.35
TNF P01375 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.33
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25855967 0.91 NLRP3 (0.65) NLRP3IL1BTNFIRAK4KCNH2
SCHEMBL25863890 0.91 NLRP3 (0.55) NLRP3IL1BTNFKCNH2
SCHEMBL25864425 0.90 NLRP3 (0.54) NLRP3IL1BTNFKCNH2
SCHEMBL25863770 0.88 NLRP3 (0.55) NLRP3IL1BTNFKCNH2
SCHEMBL25863893 0.88 NLRP3 (0.51) NLRP3IL1BTNFKCNH2
SCHEMBL25863897 0.87 NLRP3 (0.55) NLRP3IL1BTNFKCNH2
SCHEMBL25863889 0.86 NLRP3 (0.54) NLRP3IL1BTNFKCNH2
SCHEMBL25863766 0.86 NLRP3 (0.53) NLRP3IL1BTNFKCNH2
SCHEMBL25864405 0.84 NLRP3 (0.37) NLRP3IL1BTNFIRAK4
SCHEMBL25854843 0.80 NLRP3 (0.68) NLRP3IL1BTNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed