Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | GRM8 | O00222 | 2/20 | 0.95 |
| ▸ | GRM6 | O15303 | 2/20 | 0.95 |
| ▸ | GRM7 | Q14831 | 2/20 | 0.95 |
| ▸ | GRM4 | Q14833 | 2/20 | 0.95 |
| ▸ | GSR | P00390 | 2/20 | 0.95 |
| ▸ | GRIN2D | O15399 | 1/20 | 0.95 |
| ▸ | GRIN3B | O60391 | 1/20 | 0.95 |
| ▸ | CYP1A2 | P05177 | 1/20 | 0.95 |
| ▸ | GRIK1 | P39086 | 1/20 | 0.95 |
| ▸ | GRM5 | P41594 | 1/20 | 0.95 |
| ▸ | GRIA1 | P42261 | 1/20 | 0.95 |
| ▸ | GRIA2 | P42262 | 1/20 | 0.95 |
| ▸ | GRIA3 | P42263 | 1/20 | 0.95 |
| ▸ | SLC1A3 | P43003 | 1/20 | 0.95 |
| ▸ | SLC1A2 | P43004 | 1/20 | 0.95 |
| ▸ | SLC1A1 | P43005 | 1/20 | 0.95 |
| ▸ | GRIA4 | P48058 | 1/20 | 0.95 |
| ▸ | GRIN1 | Q05586 | 1/20 | 0.95 |
| ▸ | GRIN2A | Q12879 | 1/20 | 0.95 |
| ▸ | GRIK2 | Q13002 | 1/20 | 0.95 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| D-Glutamate SCHEMBL21638311 | 1.00 | GRM8 (0.95) | GRM8GRM6GRM7GRM4GSR | |
| Glutamic Acid SCHEMBL161675 | 1.00 | GRM8 (0.95) | GRM8GRM6GRM7GRM4GSR | |
| D-Glutamate SCHEMBL10427323 | 0.97 | GRM8 (0.90) | GRM8GRM6GRM7GRM4GSR | |
| Glutamic Acid SCHEMBL2826642 | 0.97 | GRM8 (0.90) | GRM8GRM6GRM7GRM4GSR | |
| D-Glutamate SCHEMBL2828267 | 0.97 | GRM8 (0.90) | GRM8GRM6GRM7GRM4GSR | |
| D-Glutamate SCHEMBL1330484 | 0.97 | GRM8 (1.00) | GRM8GRM6GRM7GRM4GSR | |
| D-Glutamate SCHEMBL1330824 | 0.97 | GRM8 (1.00) | GRM8GRM6GRM7GRM4GSR | |
| Glutamic Acid SCHEMBL1554237 | 0.97 | GRM8 (1.00) | GRM8GRM6GRM7GRM4GSR | |
| D-Glutamate SCHEMBL2201 | 0.97 | GRM8 (1.00) | GRM8GRM6GRM7GRM4GSR | |
| D-Glutamate SCHEMBL17127348 | 0.97 | GRM8 (1.00) | GRM8GRM6GRM7GRM4GSR |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 51 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-8609616-B2 | Strontium-containing compounds for use in the prevention or treatment of necrotic bone conditions | OSTEOLOGIX A/S (DK) | 2013-12-17 | — | — | US | claimed |
| EP-2266584-B1 | Composition with strontium and vitamin D for the prophylaxis and/or treatment of cartilage and/or bone conditions | OSTEOLOGIX AS (DK) | 2012-09-05 | — | — | EP | claimed |
| US-20110269675-A1 | STRONTIUM-CONTAINING COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF NECROTIC BONE CONDITIONS | OSTEOLOGIX A/S | 2011-11-03 | — | — | US | claimed |
| EP-1732575-B1 | STRONTIUM-CONTAINING COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF NECROTIC BONE CONDITIONS | OSTEOLOGIX AS (DK) | 2010-12-29 | — | — | EP | claimed |
| US-20100143473-A1 | COMBINATION TREATMENT WITH STRONTIUM FOR THE PROPHYLAXIS AND/OR TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | OSTEOLOGIX A/S | 2010-06-10 | — | — | US | claimed |
| US-7589235-B2 | High yield and rapid synthesis methods for producing metallo-organic salts | OSTEOLOGIX, A/S (DK) | 2009-09-15 | — | — | US | claimed |
| US-20080167513-A1 | Strontium-Containing Compounds for Use in the Prevention or Treatment of Necrotic Bone Conditions | OSTEOLOGLX A/S (DK) | 2008-07-10 | — | — | US | claimed |
| US-20070282127-A1 | High Yield And Rapid Synthesis Methods For Producing Metallo-Organic Salts | OSTEOLOGIX A/S | 2007-12-06 | — | — | US | claimed |
| EP-1744770-A2 | HIGH YIELD AND RAPID SYNTHESES METHODS FOR PRODUCING METALLO-ORGANIC SALTS | Osteologix A/S (DK) | 2007-01-24 | — | — | EP | claimed |
| EP-1745791-A2 | Treating cartilage/bone conditions with water-soluble strontium salts | Osteologix A/S (DK) | 2007-01-24 | — | — | EP | claimed |
| EP-1732575-A1 | STRONTIUM-CONTAINING COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF NECROTIC BONE CONDITIONS | Osteologix A/S (DK) | 2006-12-20 | — | — | EP | claimed |
| US-20060275503-A1 | Combination treatment with strontium for the prophylaxis and/or treatment of cartilage and/or bone conditions | NORDIC BONE A/S (DK) | 2006-12-07 | — | — | US | claimed |
| US-20060122274-A1 | Water-soluble strontium salts for use in treatment of cartilage and/or bone conditions | OSTEOLOGIX A/S (DK) | 2006-06-08 | — | — | US | claimed |
| EP-1622630-A2 | STRONTIUM COMBINATIONS FOR THE PROPHYLAXIS/TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | Osteologix A/S (DK) | 2006-02-08 | — | — | EP | claimed |
| WO-2005108339-A2 | HIGH YIELD AND RAPID SYNTHESES METHODS FOR PRODUCING METALLO-ORGANIC SALTS | OSTEOLOGIX A/S (DK) | 2005-11-17 | — | — | WO | claimed |
| WO-2005082385-A1 | STRONTIUM-CONTAINING COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF NECROTIC BONE CONDITIONS | OSTEOLOGIX A/S (DK) | 2005-09-09 | — | — | WO | claimed |
| EP-1534305-A2 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | Osteologix A/S (DK) | 2005-06-01 | — | — | EP | claimed |
| WO-2004098619-A2 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | OSTEOLOGIX A/S (DK) | 2004-11-18 | — | — | WO | claimed |
| WO-2004098618-A2 | STRONTIUM COMBINATIONS FOR PROPHYLAXIS/TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | OSTEOLOGIX A/S (DK) | 2004-11-18 | — | — | WO | claimed |
| US-8623422-B2 | Combination treatment with strontium for the prophylaxis and/or treatment of cartilage and/or bone conditions | OSTEOLOGIX A/S (DK) | 2014-01-07 | — | — | US | disclosed |
| US-8541471-B2 | Water-soluble strontium salts for use in treatment of cartilage and/or bone conditions | OSTEOLOGIX A/S (DK) | 2013-09-24 | — | — | US | disclosed |
| EP-1622629-B1 | Controlled-release composition containing a strontium salt | OSTEOLOGIX AS (DK) | 2013-07-10 | — | — | EP | disclosed |
| EP-1745791-B1 | Treating cartilage/bone conditions with water-soluble strontium salts | OSTEOLOGIX AS (DK) | 2013-06-26 | — | — | EP | disclosed |
| EP-2266585-B1 | Water-soluble strontium salts for use in treatment of cartilage and/or bone conditions | OSTEOLOGIX AS (DK) | 2013-06-26 | — | — | EP | disclosed |
| US-20130071496-A1 | CONTROLLED RELEASE COMPOSITION CONTAINING A STRONTIUM SALT | OSTEOLOGIX A/S (DK) | 2013-03-21 | — | — | US | disclosed |
| EP-2266584-B1 | Composition with strontium and vitamin D for the prophylaxis and/or treatment of cartilage and/or bone conditions | OSTEOLOGIX AS (DK) | 2012-09-05 | — | — | EP | disclosed |
| EP-1622630-B1 | STRONTIUM COMBINATIONS FOR THE PROPHYLAXIS/TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | OSTEOLOGIX AS (DK) | 2012-08-29 | — | — | EP | disclosed |
| US-8183409-B2 | High yield and rapid synthesis methods for producing metallo-organic salts | OSTEOLOGIX A/S (DK) | 2012-05-22 | — | — | US | disclosed |
| EP-2266584-A2 | Composition with strontium and vitamin D for the prophylaxis and/or treatment of cartilage and/or bone conditions | Osteologix A/S (DK) | 2010-12-29 | — | — | EP | disclosed |
| EP-2266585-A2 | Water-soluble strontium salts for use in treatment of cartilage and/or bone conditions | Osteologix A/S (DK) | 2010-12-29 | — | — | EP | disclosed |
| US-20100143473-A1 | COMBINATION TREATMENT WITH STRONTIUM FOR THE PROPHYLAXIS AND/OR TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | OSTEOLOGIX A/S | 2010-06-10 | — | — | US | disclosed |
| US-20100048697-A1 | WATER-SOLUBLE STRONTIUM SALTS FOR USE IN TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | HANSEN CHRISTIAN | 2010-02-25 | — | — | US | disclosed |
| US-20090291926-A1 | HIGH YIELD AND RAPID SYNTHESIS METHODS FOR PRODUCING METALLO-ORGANIC SALTS | CHRISTGAU STEPHAN | 2009-11-26 | — | — | US | disclosed |
| US-7595342-B2 | Water-soluble strontium salts for use in treatment of cartilage and/or bone conditions | OSTEOLOGIX A/S (DK) | 2009-09-29 | — | — | US | disclosed |
| US-7589235-B2 | High yield and rapid synthesis methods for producing metallo-organic salts | OSTEOLOGIX, A/S (DK) | 2009-09-15 | — | — | US | disclosed |
| US-20090191282-A1 | CONTROLLED RELEASE COMPOSITION CONTAINING A STRONTIUM SALT | OSTEOLOGIX A/S | 2009-07-30 | — | — | US | disclosed |
| US-20070282127-A1 | High Yield And Rapid Synthesis Methods For Producing Metallo-Organic Salts | OSTEOLOGIX A/S | 2007-12-06 | — | — | US | disclosed |
| EP-1534305-B9 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | OSTEOLOGIX AS (DK) | 2007-03-07 | — | — | EP | disclosed |
| EP-1744770-A2 | HIGH YIELD AND RAPID SYNTHESES METHODS FOR PRODUCING METALLO-ORGANIC SALTS | Osteologix A/S (DK) | 2007-01-24 | — | — | EP | disclosed |
| EP-1745791-A2 | Treating cartilage/bone conditions with water-soluble strontium salts | Osteologix A/S (DK) | 2007-01-24 | — | — | EP | disclosed |
| US-20060275503-A1 | Combination treatment with strontium for the prophylaxis and/or treatment of cartilage and/or bone conditions | NORDIC BONE A/S (DK) | 2006-12-07 | — | — | US | disclosed |
| EP-1534305-B1 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | OSTEOLOGIX AS (DK) | 2006-10-18 | — | — | EP | disclosed |
| US-20060216358-A1 | Controlled release composition containing a strontium salt | OSTEOLOGIX A/S (DK) | 2006-09-28 | — | — | US | disclosed |
| US-20060122274-A1 | Water-soluble strontium salts for use in treatment of cartilage and/or bone conditions | OSTEOLOGIX A/S (DK) | 2006-06-08 | — | — | US | disclosed |
| EP-1622630-A2 | STRONTIUM COMBINATIONS FOR THE PROPHYLAXIS/TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | Osteologix A/S (DK) | 2006-02-08 | — | — | EP | disclosed |
| EP-1622629-A2 | CONTROLLED RELEASE COMPOSITION CONTAINING A STRONTIUM SALT | Osteologix A/S (DK) | 2006-02-08 | — | — | EP | disclosed |
| WO-2005108339-A2 | HIGH YIELD AND RAPID SYNTHESES METHODS FOR PRODUCING METALLO-ORGANIC SALTS | OSTEOLOGIX A/S (DK) | 2005-11-17 | — | — | WO | disclosed |
| EP-1534305-A2 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | Osteologix A/S (DK) | 2005-06-01 | — | — | EP | disclosed |
| WO-2004098619-A2 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | OSTEOLOGIX A/S (DK) | 2004-11-18 | — | — | WO | disclosed |
| WO-2004098619-A2 | TREATING CARTILAGE / BONE CONDITIONS WITH WATER-SOLUBLE STRONTIUM SALTS | OSTEOLOGIX A/S (DK) | 2004-11-18 | — | — | WO | disclosed |
| WO-2004098618-A2 | STRONTIUM COMBINATIONS FOR PROPHYLAXIS/TREATMENT OF CARTILAGE AND/OR BONE CONDITIONS | OSTEOLOGIX A/S (DK) | 2004-11-18 | — | — | WO | disclosed |
| WO-2004098617-A2 | CONTROLLED RELEASE COMPOSITION CONTAINING A STRONTIUM SALT | OSTEOLOGIX A/S (DK) | 2004-11-18 | — | — | WO | disclosed |