SCHEMBL25869426

SCHEMBL25869426

CCc1nc2c(F)cc([N+](=O)[O-])cn2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 3/20 0.35
POLB P06746 4/20 0.34
HTT P42858 2/20 0.34
ALDH1A1 P00352 5/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
S1PR4 O95977 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
NFKB1 P19838 1/20 0.31
CASP3 P42574 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25311822 0.81 MAPT (0.37) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL20094248 0.72 PDE10A (0.41) LMNASMN1; SMN2CYP1A2CYP2C19NPC1
SCHEMBL25311469 0.70 ALDH1A1 (0.36) MAPTLMNAHTTALDH1A1S1PR4
SCHEMBL25309468 0.68 S1PR4 (0.39) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL25311595 0.67 MAPT (0.38) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL25311294 0.67 MAPT (0.35) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL25310974 0.65 ALDH1A1 (0.36) MAPTNPSR1LMNAPOLBHTT
SCHEMBL25312423 0.65 MAPT (0.36) MAPTLMNAHTTALDH1A1SMN1; SMN2
SCHEMBL31393110 0.64 KDM4E (0.45) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL31038494 0.64 ALDH1A1 (0.39) MAPTLMNAPOLBALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023139479-A1 SUBSTITUTED BICYCLIC HETEROCYCLES AS MALT-1 INHIBITORS AURIGENE ONCOLOGY LIMITED (IN) 2023-07-27 WO disclosed