SCHEMBL2587686

SCHEMBL2587686

CCc1c(CN2CCC2)cccc1-c1nnc(-c2ccc(CC(C)C)c(C#N)c2)s1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.60
S1PR3 Q99500 1/20 0.51
CYP2C9 P11712 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1293287 0.88 S1PR1 (0.67) S1PR1S1PR3CYP2C9
SCHEMBL1293177 0.87 S1PR1 (0.68) S1PR1S1PR3CYP2C9
SCHEMBL1293006 0.87 S1PR1 (0.68) S1PR1S1PR3CYP2C9
SCHEMBL1293335 0.87 S1PR1 (0.77) S1PR1S1PR3CYP2C9
SCHEMBL1293352 0.85 S1PR1 (0.58) S1PR1S1PR3CYP2C9
SCHEMBL12102741 0.85 S1PR1 (0.56) S1PR1S1PR3CYP2C9
SCHEMBL1293178 0.85 S1PR1 (0.70) S1PR1S1PR3CYP2C9
SCHEMBL1293331 0.85 S1PR1 (0.70) S1PR1S1PR3CYP2C9
Trifluoroacetic Acid SCHEMBL1293160 0.84 S1PR1 (0.62) S1PR1S1PR3CYP2C9
SCHEMBL1293104 0.84 S1PR1 (0.66) S1PR1S1PR3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563785-A1 COMPOUNDS AS AGONISTS OF S1P1 RECEPTORS Glaxo Group Limited (GB) 2013-03-06 EP disclosed
WO-2011134280-A1 COMPOUNDS AS AGONISTS OF S1P1 RECEPTORS GLAXO GROUP LIMITED (GB) 2011-11-03 WO disclosed