SCHEMBL2587965

SCHEMBL2587965

S=P(c1ccccc1)(c1ccccc1)c1cnc2ccccn12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 8/20 1.00
FLT3 P36888 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
GPR84 Q9NQS5 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
GGPS1 O95749 1/20 0.39
FDPS P14324 1/20 0.39
MIF P14174 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.38
PKM P14618 1/20 0.38
EPHB3 P54753 1/20 0.38
GAA P10253 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590640 0.81 NPSR1 (0.69) NPSR1FLT3NPC1RAB9AGPR84
SCHEMBL23132987 0.70 NPSR1 (0.53) NPSR1FLT3NPC1RAB9AGPR84
SCHEMBL14756611 0.68 NPC1 (0.53) NPSR1FLT3NPC1RAB9AGPR84
SCHEMBL496758 0.68 NPC1 (0.60) NPSR1NPC1RAB9AADORA3GGPS1
SCHEMBL2650330 0.67 FLT3 (0.74) NPSR1FLT3MIFIRAK4PKM
SCHEMBL2582202 0.67 NPSR1 (1.00) NPSR1NPC1GAAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL21834227 0.67 NPC1 (0.59) NPSR1NPC1RAB9AADORA3GGPS1
SCHEMBL31734376 0.67 NPC1 (0.51) NPSR1FLT3NPC1RAB9AADORA3
SCHEMBL504102 0.66 NPSR1 (0.50) NPSR1FLT3NPC1RAB9AADORA3
SCHEMBL3313454 0.66 MIF (0.53) NPSR1FLT3NPC1RAB9AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137220-A1 SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-11-03 WO disclosed
WO-2011137220-A1 SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-11-03 WO disclosed