SCHEMBL25879887

SCHEMBL25879887

CNC(=O)c1cc(Nc2ncc3c(CNC(=O)c4cc(Nc5ncc6ccc(-c7cn[nH]c7)cc6n5)c[nH]4)cc(Br)cc3n2)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.42
MAP3K5 Q99683 2/20 0.41
JUN P05412 2/20 0.39
MAPK10 P53779 2/20 0.39
ROCK2 O75116 13/20 0.37
ROCK1 Q13464 10/20 0.37
MAPK8 P45983 1/20 0.37
PRKACA P17612 1/20 0.36
PRKACG P22612 1/20 0.36
PRKACB P22694 1/20 0.36
USP30 Q70CQ3 1/20 0.34
BRAF P15056 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512127 0.85 MAP3K5 (0.53) MAP4K1MAP3K5JUNMAPK10ROCK2
SCHEMBL25881300 0.85 MAP3K5 (0.53) MAP4K1MAP3K5JUNMAPK10ROCK2
SCHEMBL25882124 0.79 MAP3K5 (0.63) MAP4K1MAP3K5ROCK2ROCK1BRAF
SCHEMBL25881895 0.78 CREBBP (0.46) MAP3K5BRAF
SCHEMBL25879716 0.77 PTK2 (0.39)
SCHEMBL25881914 0.75 MAP3K5 (0.52) MAP4K1MAP3K5JUNMAPK10ROCK2
SCHEMBL30512125 0.74 MAP4K1 (0.59) MAP4K1MAP3K5JUNMAPK10ROCK2
SCHEMBL30512117 0.72 MAP4K1 (0.41) MAP4K1MAP3K5JUNMAPK10BRAF
SCHEMBL25882103 0.72 MAP4K1 (0.41) MAP4K1MAP3K5JUNMAPK10BRAF
SCHEMBL30512131 0.72 MAP3K5 (0.61) MAP4K1MAP3K5JUNMAPK10ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed