SCHEMBL25880620

SCHEMBL25880620

CNC(=O)c1cc(Nc2ncc3ccc(-c4cnn(CNC(=O)c5cc(Nc6ncc7cc(-c8cn[nH]c8)ccc7n6)c[nH]5)c4)cc3n2)sn1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 2/20 0.42
MAP4K1 Q92918 4/20 0.39
JUN P05412 2/20 0.36
MAPK10 P53779 2/20 0.36
BRAF P15056 9/20 0.34
MAPK8 P45983 1/20 0.34
RAF1 P04049 1/20 0.34
TTK P33981 1/20 0.34
ROCK2 O75116 1/20 0.33
PTK6 Q13882 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512123 0.81 MAP4K1 (0.49) MAP3K5MAP4K1JUNMAPK10BRAF
SCHEMBL25882177 0.81 MAP4K1 (0.49) MAP3K5MAP4K1JUNMAPK10BRAF
SCHEMBL25880784 0.81 MAP3K5 (0.55) MAP3K5MAP4K1BRAFROCK2PTK6
SCHEMBL25882124 0.77 MAP3K5 (0.63) MAP3K5MAP4K1BRAFRAF1ROCK2
SCHEMBL25881300 0.77 MAP3K5 (0.53) MAP3K5MAP4K1JUNMAPK10BRAF
SCHEMBL30512127 0.77 MAP3K5 (0.53) MAP3K5MAP4K1JUNMAPK10BRAF
SCHEMBL25879887 0.70 MAP4K1 (0.42) MAP3K5MAP4K1JUNMAPK10BRAF
SCHEMBL25881914 0.69 MAP3K5 (0.52) MAP3K5MAP4K1JUNMAPK10MAPK8
SCHEMBL30512125 0.68 MAP4K1 (0.59) MAP3K5MAP4K1JUNMAPK10BRAF
SCHEMBL30512131 0.66 MAP3K5 (0.61) MAP3K5MAP4K1JUNMAPK10BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed