SCHEMBL2588127

SCHEMBL2588127

NS(=O)(=O)c1cccc(-c2n[nH]c3ccc(NC(=O)Cc4cccs4)cc23)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TTK P33981 19/20 1.00
PLK4 O00444 1/20 0.62
CHEK2 O96017 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
AURKB Q96GD4 1/20 0.62
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA5A P35218 1/20 0.58
CA7 P43166 1/20 0.58
CA9 Q16790 1/20 0.58
CA13 Q8N1Q1 1/20 0.58
CA5B Q9Y2D0 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12281383 0.92 TTK (0.85) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL12282318 0.87 TTK (1.00) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL2861303 0.86 TTK (0.75) TTKAURKB
SCHEMBL2569400 0.86 TTK (1.00) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL2571823 0.85 TTK (0.78) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL2570870 0.85 TTK (1.00) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL12281036 0.85 TTK (0.80) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL12284278 0.83 TTK (1.00) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL12284538 0.83 TTK (0.84) TTKPLK4CHEK2CYP3A4CYP2C9
SCHEMBL2564623 0.83 TTK (1.00) TTKPLK4CHEK2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed