SCHEMBL25890286

SCHEMBL25890286

CC1(O)C(=O)N(c2cncc(Cc3n[nH]c(=O)c4ccccc34)c2)c2ccc(F)cc21

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.47
AR P10275 1/20 0.41
ENPP1 P22413 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25890288 1.00 PARP1 (0.47) PARP1ARENPP1CYP3A4CYP2C9
SCHEMBL30132752 0.94 PARP1 (0.40) PARP1
SCHEMBL25312643 0.94 PARP1 (0.40) PARP1
SCHEMBL25890284 0.94 PARP1 (0.40) PARP1
SCHEMBL25890291 0.93 PARP1 (0.47) PARP1ARCYP3A4CYP2C9TSHR
SCHEMBL30132743 0.91 PARP1 (0.43) PARP1AR
SCHEMBL25312615 0.91 PARP1 (0.43) PARP1AR
SCHEMBL29565341 0.91 PARP1 (0.43) PARP1AR
SCHEMBL25315024 0.91 PARP1 (0.43) PARP1AR
SCHEMBL25890280 0.91 PARP1 (0.43) PARP1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115485271-A Novel compounds as inhibitors of poly (ADP-ribose) polymerase (PARP) 理森制药股份公司 2022-12-16 CN disclosed