SCHEMBL25896262

SCHEMBL25896262

Nc1ccc(N2C[C@@H]3C[C@H]2CN3CCF)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 3/20 0.44
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
PIK3CD O00329 1/20 0.32
MAP3K12 Q12852 2/20 0.31
BRAF P15056 1/20 0.31
ALDH1A1 P00352 2/20 0.31
MAPT P10636 2/20 0.31
GFER P55789 2/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
ADRA2C P18825 1/20 0.31
KMT2A Q03164 1/20 0.31
PTK2B Q14289 1/20 0.31
ESR2 Q92731 1/20 0.31
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24680997 0.85 DRD3 (0.58) DRD3DRD2DRD4PIK3CDHDAC1
SCHEMBL2718724 0.85 DRD3 (0.44) DRD3DRD2DRD4MAP3K12BRAF
SCHEMBL24680998 0.85 DRD3 (0.58) DRD3DRD2DRD4PIK3CDHDAC1
SCHEMBL5493145 0.77 HDAC1 (0.46) DRD3DRD2DRD4MAPTHDAC1
SCHEMBL2729685 0.76 KCNH2 (0.44) BRAFALDH1A1MAPTGFERKDM4E
SCHEMBL21641736 0.76 KCNH2 (0.44) BRAFALDH1A1MAPTGFERKDM4E
SCHEMBL5497644 0.73 DRD3 (0.58) DRD3DRD2DRD4HDAC1AKR1C3
SCHEMBL2391102 0.69 KDM4E (0.33) ALDH1A1MAPTGFERHTTKDM4E
SCHEMBL1898615 0.69 MAP3K12 (0.42) MAP3K12ALDH1A1MAPTGFERHTT
SCHEMBL19381939 0.69 DRD3 (0.44) DRD3DRD2DRD4MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138362-A1 WEE1 INHIBITOR, PREPARATION THEREFOR, AND USE THEREOF 江苏天士力帝益药业有限公司 2023-07-27 WO disclosed