SCHEMBL2590109

SCHEMBL2590109

COC(C)Cn1ccc(C(=O)O)cc1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
B3GNT2 Q9NY97 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA7 P43166 1/20 0.36
TPMT P51580 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
KDM4E B2RXH2 3/20 0.35
HCAR3 P49019 1/20 0.35
ACACB O00763 2/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 1/20 0.34
TSHR P16473 1/20 0.34
POLB P06746 1/20 0.34
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29168986 0.82 HTR2C (0.41) B3GNT2KMT2A
SCHEMBL29168988 0.82 HTR2C (0.41) B3GNT2KMT2A
SCHEMBL13522485 0.76 B3GNT2 (0.35) B3GNT2ALDH1A1KDM4EACACBKMT2A
SCHEMBL4246332 0.76 POLB (0.47) ALDH1A1KDM4EHCAR3ACACBKMT2A
SCHEMBL2583269 0.76 ALDH1A1 (0.54) ALDH1A1CA12CA1CA2CA4
SCHEMBL1015082 0.75 ALDH1A1 (0.46) ALDH1A1CA12CA1CA2CA7
SCHEMBL29169219 0.74 ACACB (0.36) CA1CA2CA4CA7CA9
SCHEMBL29169222 0.74 ACACB (0.36) CA1CA2CA4CA7CA9
SCHEMBL16417103 0.74 LPAR1 (0.42) CA12CA1CA2CA4CA6
SCHEMBL13522486 0.73 ALDH1A1 (0.48) ALDH1A1HCAR3ACACBHTTKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595989-A1 HETEROCYCLIC CHROMENE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS Vertex Pharmaceuticals Incorporated (US) 2013-05-29 EP disclosed
WO-2013067248-A1 BENZOXAZINES AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-05-10 WO disclosed
WO-2011140425-A1 HETEROCYCLIC CHROMENE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-10 WO disclosed