SCHEMBL2592356

SCHEMBL2592356

COn1c(C=O)cc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.46
CYP2A6 P11509 1/20 0.38
MAOA P21397 2/20 0.36
ALDH1A1 P00352 2/20 0.36
DAO P14920 1/20 0.35
MCL1 Q07820 1/20 0.35
GAA P10253 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
ERN1 O75460 1/20 0.34
KMT2A Q03164 1/20 0.33
BACE1 P56817 1/20 0.33
PTGER4 P35408 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5642556 0.84 SMN1; SMN2 (0.42) SMN1; SMN2CYP2A6MAOAALDH1A1DAO
SCHEMBL8932716 0.76 CNR2 (0.33) SMN1; SMN2MAOAGAAKMT2ACYP1A2
SCHEMBL29894136 0.76 GRIN2D (0.51) ALDH1A1DAOMCL1GRIN2DGRIN3B
SCHEMBL342762 0.76 GRIN2D (0.51) ALDH1A1DAOMCL1GRIN2DGRIN3B
SCHEMBL4784169 0.75 PTGER4 (0.43) SMN1; SMN2CYP2A6ALDH1A1KMT2APTGER4
SCHEMBL21803766 0.75 KDM4E (0.41) SMN1; SMN2CYP2A6ALDH1A1GRIN2DGRIN3B
SCHEMBL30229435 0.73 PTGER4 (0.55) SMN1; SMN2ALDH1A1GAAKMT2APTGER4
SCHEMBL18247464 0.73 PTGER4 (0.55) SMN1; SMN2ALDH1A1GAAKMT2APTGER4
SCHEMBL670199 0.73 SMN1; SMN2 (0.47) SMN1; SMN2CYP2A6ALDH1A1DAOMCL1
SCHEMBL4589923 0.73 CYP2A6 (0.42) CYP2A6ALDH1A1DAOMCL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011139242-A2 PROCESS FOR THE PREPARATION OF 2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLE DERIVATIVES USTAV EXPIREMENTÁLNEJ FARMAKOLÓGIE A TOXIKOLÓGIE SAV (SK) 2011-11-10 WO disclosed