SCHEMBL2592425

SCHEMBL2592425

CN(Cc1ccccc1)c1nc(-c2ccc([N+](=O)[O-])cc2)nc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 1.00
CYP1A2 P05177 4/20 1.00
POLB P06746 3/20 1.00
NPSR1 Q6W5P4 3/20 1.00
CYP3A4 P08684 3/20 1.00
CYP2C9 P11712 3/20 1.00
ALDH1A1 P00352 5/20 0.78
PDE5A O76074 1/20 0.73
ABCG2 Q9UNQ0 4/20 0.66
KMT2A Q03164 4/20 0.58
MEN1 O00255 3/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
LMNA P02545 3/20 0.58
MCL1 Q07820 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
GBA1 P04062 3/20 0.56
NPC1 O15118 1/20 0.54
XBP1 P17861 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590347 0.88 ALDH1A1 (1.00) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL1085047 0.85 PDE5A (1.00) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL4084599 0.82 PDE5A (0.82) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL4090063 0.80 PDE5A (0.78) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL4095681 0.76 PDE5A (0.72) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL12175988 0.76 POLB (0.61) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL28797852 0.76 NPSR1 (0.65) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL1083881 0.75 PDE5A (0.78) MAPTCYP1A2POLBNPSR1CYP3A4
SCHEMBL18353944 0.75 GBA1 (0.93) MAPTCYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL15289676 0.74 POLB (0.98) MAPTCYP1A2POLBNPSR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed