Formic Acid

Formic Acid

SCHEMBL2592575

C[C@@]1(c2cc(NC(=O)c3ccc(Cl)cn3)ccc2F)CCOCC(N)=N1.O=CO

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.93
BACE2 Q9Y5Z0 2/20 0.72
CTSD P07339 2/20 0.66
APP P05067 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584678 0.96 BACE1 (1.00) BACE1BACE2CTSDAPP
SCHEMBL7702958 0.89 BACE1 (0.86) BACE1BACE2CTSDAPP
SCHEMBL1173499 0.87 BACE1 (1.00) BACE1APP
SCHEMBL360663 0.87 BACE1 (1.00) BACE1APP
SCHEMBL16509555 0.85 BACE1 (0.84) BACE1BACE2
SCHEMBL2588794 0.85 BACE1 (0.84) BACE1BACE2APP
SCHEMBL2587828 0.85 BACE1 (0.78) BACE1BACE2APP
Formic Acid SCHEMBL2592659 0.84 BACE1 (0.67) BACE1BACE2APP
SCHEMBL15703749 0.84 BACE1 (0.77) BACE1BACE2CTSD
SCHEMBL1975402 0.84 BACE1 (1.00) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138293-A1 2,5,6,7-TETRAHYDRO-[1,4]OXAZEPIN-3-YLAMINE OR 2,3,6,7-TETRAHYDRO-[1,4]OXAZEPIN-5-YLAMINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-11-10 WO disclosed