SCHEMBL25928142

SCHEMBL25928142

O=C(Nc1sc2ccccc2c1Br)c1ccc(-c2nc3ccccc3n2-c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
SCD O00767 1/20 0.43
PTGER4 P35408 1/20 0.42
ADORA1 P30542 1/20 0.42
RECQL P46063 1/20 0.41
EGFR P00533 1/20 0.41
SIRT2 Q8IXJ6 2/20 0.41
SIRT1 Q96EB6 2/20 0.41
GRIA1 P42261 1/20 0.40
CACNG8 Q8WXS5 1/20 0.40
CACNG2 Q9Y698 1/20 0.40
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25929182 0.80 HDAC6 (0.42) HDAC1HDAC6ALDH1A1CASP3SENP7
SCHEMBL25927553 0.79 HDAC1 (0.44) ADORA3HDAC1HDAC8HDAC6ESR1
SCHEMBL18347069 0.76 EGFR (0.46) ADORA3HDAC1HDAC8HDAC6ESR1
SCHEMBL17343544 0.74 HDAC1 (0.45) HDAC1HDAC8HDAC6ESR1ESR2
SCHEMBL21760739 0.74 ESR1 (0.62) HDAC1HDAC8HDAC6ESR1ESR2
SCHEMBL713654 0.73 ESR1 (0.56) HDAC1HDAC8HDAC6ESR1ESR2
SCHEMBL21760742 0.73 ESR1 (0.61) HDAC1HDAC8HDAC6ESR1ESR2
SCHEMBL25928110 0.72 HDAC6 (0.56) HDAC6SCDALDH1A1NPC1RAB9A
SCHEMBL17343543 0.72 ESR1 (0.59) HDAC1HDAC8HDAC6ESR1ESR2
SCHEMBL25927861 0.72 KMT2A (0.57) HDAC1HDAC8HDAC6ALDH1A1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138254-A1 HETEROCYCLIC COMPOUND, AND ORGANIC ELECTROLUMINESCENT MATERIAL AND ELEMENT 上海八亿时空先进材料有限公司 2023-07-27 WO disclosed