SCHEMBL25930863

SCHEMBL25930863

Cc1cc(Br)cnc1N1C[C@@H](C)O[C@H](C)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
HSD17B10 Q99714 3/20 0.40
TSHR P16473 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 8/20 0.40
GAA P10253 3/20 0.40
HTT P42858 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
POLB P06746 1/20 0.39
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
LMNA P02545 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ATM Q13315 1/20 0.38
RAB9A P51151 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25930953 1.00 KDM4E (0.40) KDM4EHSD17B10TSHRNPSR1ALDH1A1
SCHEMBL25929001 0.83 OPRK1 (0.40) MTOR
SCHEMBL29173621 0.82 LRRK2 (0.43)
SCHEMBL30205934 0.82 LRRK2 (0.43)
SCHEMBL29209035 0.81 PIK3CA (0.43) KDM4EHSD17B10TSHRNPSR1ALDH1A1
SCHEMBL29209033 0.81 PIK3CA (0.43) KDM4EHSD17B10TSHRNPSR1ALDH1A1
SCHEMBL29208999 0.81 PIK3CA (0.43) KDM4EHSD17B10TSHRNPSR1ALDH1A1
SCHEMBL18483979 0.81 OPRK1 (0.40)
SCHEMBL25931749 0.80 OPRK1 (0.42)
SCHEMBL2214488 0.80 OPRK1 (0.48) KDM4EALDH1A1GAAHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131271-A1 PYRROLE FUSED-RING PYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 杭州中美华东制药有限公司 2023-07-13 WO disclosed