SCHEMBL25933757

SCHEMBL25933757

NCc1csc(C2(c3cccc(Cl)c3)CCOCC2)n1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2RL3 Q96RI0 10/20 0.44
SLC6A4 P31645 3/20 0.39
SLC6A3 Q01959 3/20 0.39
ICMT O60725 1/20 0.37
HTR2C P28335 2/20 0.37
HTR2A P28223 1/20 0.37
HTR2B P41595 1/20 0.37
DPP4 P27487 3/20 0.34
DPP9 Q86TI2 2/20 0.33
DPP8 Q6V1X1 1/20 0.33
SLC6A2 P23975 2/20 0.32
PNMT P11086 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15349057 0.88 F2RL3 (0.44) F2RL3SLC6A4SLC6A3ICMTHTR2C
SCHEMBL25933735 0.86 F2RL3 (0.42) F2RL3SLC6A4SLC6A3SLC6A2
SCHEMBL15349224 0.83 F2RL3 (0.46) F2RL3SLC6A4SLC6A3ICMTSLC6A2
SCHEMBL15349123 0.74 F2RL3 (0.42) F2RL3
SCHEMBL15349106 0.72 F2RL3 (0.39) F2RL3
SCHEMBL15348977 0.71 F2RL3 (0.49) F2RL3ICMT
SCHEMBL15057062 0.69 SLC6A4 (0.71) SLC6A4SLC6A3ICMTDPP4DPP9
SCHEMBL25933755 0.69 ICMT (0.38) F2RL3SLC6A4SLC6A3ICMTSLC6A2
Hydrochloric Acid SCHEMBL29428954 0.68 SLC6A4 (0.69) SLC6A4SLC6A3ICMTHTR2CHTR2A
SCHEMBL5646704 0.68 ROCK1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242535-A1 IMIDAZOTHIADIAZOLE AND IMIDAZOPYRAZINE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION BRISTOL MYERS SQUIBB CO (US) 2023-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242535-A1 IMIDAZOTHIADIAZOLE AND IMIDAZOPYRAZINE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION F2RL3, F2R, TMPRSS4 F2RL3 1/4885SLC6A4 413/4885SLC6A3 1513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.