SCHEMBL2594720

SCHEMBL2594720

COc1ccc2c(c1)C(=O)CC1(CCN(C(=O)O)CC1)O2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.59
KDM4E B2RXH2 11/20 0.59
GAA P10253 6/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
HPGD P15428 8/20 0.58
CASP1 P29466 6/20 0.58
HSD17B10 Q99714 6/20 0.58
GLA P06280 6/20 0.57
CASP7 P55210 3/20 0.57
KMT2A Q03164 2/20 0.57
CYP1A2 P05177 1/20 0.57
THRB P10828 1/20 0.55
CYP19A1 P11511 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA7 P43166 1/20 0.54
CA9 Q16790 1/20 0.54
KLK7 P49862 1/20 0.54
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567882 0.88 HDAC3 (0.68) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL13005009 0.86 KDM4E (0.60) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL4258170 0.85 KMT2A (0.57) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL14433515 0.85 ALDH1A1 (0.57) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL620146 0.83 KDM4E (0.63) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL732843 0.83 HDAC3 (0.64) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL13791467 0.82 CA1 (0.63) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL9444279 0.82 KDM4E (0.68) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL731330 0.82 KMT2A (0.53) ALDH1A1KDM4EGAASMN1; SMN2HPGD
SCHEMBL308831 0.81 KMT2A (0.57) ALDH1A1KDM4EGAASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595989-A1 HETEROCYCLIC CHROMENE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS Vertex Pharmaceuticals Incorporated (US) 2013-05-29 EP disclosed
WO-2011140425-A1 HETEROCYCLIC CHROMENE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-10 WO disclosed