SCHEMBL25947832

SCHEMBL25947832

O=C/C=C/CCCC(=O)Nc1cccn(Cc2cc3ccccc3[nH]2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MAP4K1 Q92918 11/20 0.42
HDAC3 O15379 4/20 0.40
HDAC1 Q13547 4/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC8 Q9BY41 3/20 0.40
KDM4E B2RXH2 2/20 0.39
APP P05067 1/20 0.37
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
CASP1 P29466 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25939365 0.84 MAP4K1 (0.54) ALDH1A1TSHRHSD17B10MAP4K1KDM4E
SCHEMBL25944756 0.83 MAP4K1 (0.57) ALDH1A1TSHRHSD17B10MAP4K1KDM4E
SCHEMBL25945185 0.81 MAP4K1 (0.58) ALDH1A1TSHRHSD17B10MAP4K1HDAC3
SCHEMBL25945823 0.80 MAP4K1 (0.40) ALDH1A1TSHRHSD17B10MAP4K1KDM4E
SCHEMBL25944422 0.78 MAP4K1 (0.57) ALDH1A1TSHRHSD17B10MAP4K1HDAC3
SCHEMBL25945112 0.78 MAP4K1 (0.57) MAP4K1
SCHEMBL25938538 0.78 MAP4K1 (0.58) ALDH1A1TSHRHSD17B10MAP4K1KDM4E
SCHEMBL25944432 0.76 MAP4K1 (0.70) MAP4K1
SCHEMBL25940979 0.76 MAP4K1 (0.44) ALDH1A1TSHRHSD17B10MAP4K1KDM4E
SCHEMBL25944411 0.75 MAP4K1 (0.69) MAP4K1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4219460-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS Sitari Pharma, Inc. (US) 2023-08-02 EP disclosed