SCHEMBL2595552

SCHEMBL2595552

Cn1cc(P(=S)(c2ccccc2)c2ccccc2)[n+]2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 19/20 0.54
PSMD14 O00487 1/20 0.43
RAD52 P43351 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CHRM2 P08172 2/20 0.40
CHRM4 P08173 2/20 0.40
CHRM5 P08912 2/20 0.40
ADRA2A P08913 2/20 0.40
CHRM1 P11229 2/20 0.40
ADRB3 P13945 2/20 0.40
ADRA2C P18825 2/20 0.40
CHRM3 P20309 2/20 0.40
S1PR1 P21453 2/20 0.40
FPR1 P21462 2/20 0.40
SLC6A2 P23975 2/20 0.40
HRH2 P25021 2/20 0.40
FPR3 P25089 2/20 0.40
HTR2A P28223 2/20 0.40
AGTR1 P30556 2/20 0.40
GPR183 P32249 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2594343 0.70 NPSR1 (1.00) NPSR1PSMD14RAD52CHRM2CHRM4
SCHEMBL517954 0.60 ESR1 (0.68) NPSR1L3MBTL1
SCHEMBL12175482 0.58 NPSR1 (1.00) NPSR1HTR2A
SCHEMBL9772833 0.58 ESR1 (0.65) NPSR1L3MBTL1
SCHEMBL31176947 0.58 ESR1 (0.65) NPSR1L3MBTL1
Phosphine SCHEMBL15190577 0.58 ESR1 (0.65) NPSR1L3MBTL1
SCHEMBL8630054 0.55 ESR1 (0.42) NPSR1L3MBTL1
SCHEMBL6832368 0.54 ESR1 (0.46) NPSR1L3MBTL1
SCHEMBL7900827 0.54 ESR1 (0.46) NPSR1L3MBTL1
SCHEMBL7200128 0.54 ESR1 (0.46) NPSR1L3MBTL1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137220-A1 SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-11-03 WO disclosed