SCHEMBL2596705

SCHEMBL2596705

CCc1cc(-c2nnc(S)n2-c2ccc(OC)c3[nH]c(C(C)C)cc23)c(O)cc1O.[NaH].[NaH]

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
GAA P10253 2/20 0.33
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.30
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL788553 0.99 MEN1 (0.33) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL1586236 0.91 ALDH1A1 (0.33) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL1586624 0.89 GAA (0.33) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL1586062 0.87 HSP90AA1 (0.38) HSP90AA1
SCHEMBL1586050 0.84
SCHEMBL930136 0.82 MEN1 (0.36) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL13280018 0.81 DAO (0.34) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL445551 0.80 MEN1 (0.32) MEN1KMT2AGAA
SCHEMBL977473 0.79 MEN1 (0.35) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL421149 0.79 MEN1 (0.32) MEN1KMT2AGAAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO claimed