SCHEMBL25972793

SCHEMBL25972793

CC1(C)c2ccccc2-c2c1cc(-c1c3ccccc3c(-c3cccc4[nH]c5ccccc5c34)c3ccccc13)c1ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.39
IMPDH2 P12268 1/20 0.39
IMPDH1 P20839 1/20 0.39
CHEK1 O14757 1/20 0.35
GABRP O00591 2/20 0.35
GABRD O14764 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRB1 P18505 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35
GABRA4 P48169 2/20 0.35
GABRE P78334 2/20 0.35
GABRA6 Q16445 2/20 0.35
GABRG1 Q8N1C3 2/20 0.35
GABRG3 Q99928 2/20 0.35
GABRQ Q9UN88 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25972541 0.86 PARP1 (0.38) PARP1IMPDH2IMPDH1CHEK1GABRP
SCHEMBL25972391 0.82 AHR (0.38) PARP1GABRPGABRDGABRA1GABRB1
SCHEMBL15940475 0.80 PARP1 (0.39) PARP1IMPDH2IMPDH1CHEK1CDK4
SCHEMBL17484091 0.79 PARP1 (0.50) PARP1IMPDH2IMPDH1CHEK1GABRP
SCHEMBL29438556 0.79 PARP1 (0.50) PARP1IMPDH2IMPDH1CHEK1GABRP
SCHEMBL17998759 0.77 PARP1 (0.40) PARP1IMPDH2IMPDH1GABRPGABRD
SCHEMBL30985271 0.77 PARP1 (0.40) PARP1IMPDH2IMPDH1GABRPGABRD
SCHEMBL24004226 0.77 PGR (0.33) KDM4EMEN1MAPTKMT2AAHR
SCHEMBL20438138 0.76 PARP1 (0.45) PARP1IMPDH2IMPDH1CHEK1GABRP
SCHEMBL18687885 0.76 PARP1 (0.42) PARP1IMPDH2IMPDH1CHEK1GABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230255102-A1 PLURALITY OF HOST MATERIALS AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING THE SAME DUPONT SPECIALTY MATERIALS KOREA LTD. (KR) 2023-08-10 US disclosed