SCHEMBL25976602

SCHEMBL25976602

C=CC(=O)N1CCc2sc(C)nc2C1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.50
GRM5 P41594 3/20 0.39
EGFR P00533 8/20 0.37
DPP4 P27487 2/20 0.35
DPP8 Q6V1X1 2/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
BTK Q06187 2/20 0.33
RYR2 Q92736 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25976511 0.89 MAPK1 (0.57) MAPK1GRM5EGFRDPP4DPP8
SCHEMBL14907170 0.78 GRM5 (0.40) GRM5DPP4DPP8DPP9DPP7
SCHEMBL16219073 0.78 GRM5 (0.42) GRM5DPP4DPP8DPP9DPP7
SCHEMBL27327040 0.75 ADORA1 (0.48) GRM5
SCHEMBL25976604 0.71 MAPK1 (0.44) MAPK1GRM5BTKRYR2ACHE
SCHEMBL26032624 0.71 MAPK1 (0.47) MAPK1EGFRDPP4DPP8DPP9
SCHEMBL25976509 0.70 MAPK1 (0.46) MAPK1BTKRYR2ACHE
SCHEMBL9382117 0.70 GRM5 (0.56) GRM5DPP4DPP8DPP9DPP7
SCHEMBL8277491 0.70 HRH3 (0.48) GRM5NPC1RAB9A
SCHEMBL21452307 0.70 GRM5 (0.37) GRM5DPP4DPP8DPP9DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154282-A1 COMPOUNDS HAVING A T-STRUCTURE FORMED BY AT LEAST FOUR CYCLES FOR USE IN THE TREATMENT OF CANCER AND OTHER INDICATIONS THERAS, INC. (US) 2023-08-17 WO disclosed