SCHEMBL2598348

SCHEMBL2598348

COc1ccc(Cn2ncc3ncccc32)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.55
GRIN2B Q13224 6/20 0.55
CNR2 P34972 2/20 0.48
CNR1 P21554 1/20 0.48
NPBWR1 P48145 8/20 0.48
MCHR1 Q99705 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HKDC1 Q2TB90 1/20 0.43
PTK2 Q05397 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31513725 0.82 RECQL (0.60) GRIN1GRIN2BKDM4EALDH1A1SMN1; SMN2
SCHEMBL23210845 0.82 GRIN1 (0.61) GRIN1GRIN2BNPBWR1MCHR1
SCHEMBL28345671 0.81 RECQL (0.44) GRIN1GRIN2BALDH1A1
SCHEMBL23210996 0.78 GRIN1 (0.58) GRIN1GRIN2BNPBWR1
SCHEMBL27717175 0.78 RECQL (0.69) GRIN1GRIN2BCNR2CNR1NPBWR1
SCHEMBL22892720 0.78 NPBWR1 (0.51) GRIN1GRIN2BCNR2NPBWR1MCHR1
SCHEMBL17395029 0.78 NPBWR1 (0.48) NPBWR1MCHR1KDM4EALDH1A1LMNA
SCHEMBL30803766 0.77 GRIN1 (0.58) GRIN1GRIN2BKDM4EALDH1A1
SCHEMBL29545049 0.76 NPBWR1 (0.46) GRIN1GRIN2BCNR2CNR1NPBWR1
SCHEMBL2598351 0.76 NPBWR1 (0.49) GRIN1GRIN2BCNR2CNR1NPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146287-A1 PYRAZOLO[4,3-B]PYRIDINE-7-AMINE INHIBITORS OF ALK5 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-11-24 WO disclosed