SCHEMBL2598843

SCHEMBL2598843

O=C1NC[C@@H]2CNCC2c2ccc(-c3cccc(CCO)c3)cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 1/20 0.39
BACE1 P56817 1/20 0.37
CDK8 P49336 1/20 0.34
MAP4K4 O95819 1/20 0.34
CLK4 Q9HAZ1 2/20 0.33
DYRK1B Q9Y463 2/20 0.33
FYN P06241 1/20 0.33
TYRO3 Q06418 1/20 0.33
NTRK2 Q16620 1/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
SLC5A1 P13866 5/20 0.32
PARP1 P09874 3/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
CCNK O75909 1/20 0.31
CDK7 P50613 1/20 0.31
CCNH P51946 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1805585 1.00 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
SCHEMBL2598841 1.00 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
SCHEMBL1805583 1.00 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
Hydrochloric Acid SCHEMBL2598913 0.99 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
Hydrochloric Acid SCHEMBL1806102 0.99 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
Hydrochloric Acid SCHEMBL2598911 0.99 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
Hydrochloric Acid SCHEMBL1806104 0.99 ACMSD (0.39) ACMSDBACE1CDK8MAP4K4CLK4
SCHEMBL860924 0.83 BACE1 (0.41) ACMSDBACE1CDK8MAP4K4CLK4
SCHEMBL860923 0.83 BACE1 (0.41) ACMSDBACE1CDK8MAP4K4CLK4
SCHEMBL861233 0.82 BACE1 (0.41) ACMSDBACE1SLC5A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571353-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF AbbVie Inc. (US) 2013-03-27 EP disclosed
WO-2011146089-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2011-11-24 WO disclosed