SCHEMBL2599665

SCHEMBL2599665

COc1cccc(Oc2cnc(N3CCOc4c(F)cccc43)nc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HSD17B10 Q99714 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
BRCA1 P38398 1/20 0.38
HBB P68871 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR6 P50406 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
AVPR1A P37288 1/20 0.36
TSHR P16473 3/20 0.36
MAPK1 P28482 2/20 0.36
LMNA P02545 1/20 0.36
DCK P27707 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP17A1 P05093 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL16332340 0.94 CYP17A1 (0.36) PIK3CDPIK3CBPIK3CGALDH1A1HSD17B10
SCHEMBL2599612 0.87 PIK3CD (0.36) PIK3CDPIK3CBPIK3CGALDH1A1HTR6
SCHEMBL2599637 0.86 APP (0.41) PIK3CDPIK3CBPIK3CGHTR6AVPR1A
Dimethylamine SCHEMBL2599639 0.86 CYP17A1 (0.40) PIK3CDPIK3CBPIK3CGALDH1A1KMT2A
SCHEMBL2599603 0.85 MAPT (0.40) PIK3CDPIK3CBPIK3CGKMT2ATSHR
SCHEMBL2599623 0.84 DHFR (0.40) ALDH1A1HSD17B10KDM4EKMT2AHTR6
SCHEMBL16388793 0.82 PIK3CA (0.37) PIK3CDPIK3CBPIK3CGAVPR1ACYP1A2
SCHEMBL2599667 0.82 AVPR1A (0.35) PIK3CDPIK3CBPIK3CGHTR6AVPR1A
SCHEMBL16332713 0.81 CYP17A1 (0.34) PIK3CDPIK3CBPIK3CGHTR6AVPR1A
SCHEMBL16388603 0.80 F10 (0.37) PIK3CDPIK3CBPIK3CGAVPR1ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP claimed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP claimed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO claimed
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed