SCHEMBL26009583

SCHEMBL26009583

CN1CCN(c2cc3nccn3c(Nc3cc[nH]n3)n2)CC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.35
AURKB Q96GD4 3/20 0.35
EGFR P00533 1/20 0.35
MAPKAPK5 Q8IW41 1/20 0.35
HRH4 Q9H3N8 4/20 0.34
HRH3 Q9Y5N1 1/20 0.34
NTRK1 P04629 1/20 0.34
HTR3A P46098 2/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26009808 0.87 ATR (0.40) MAPKAPK5
SCHEMBL3042183 0.83 AURKA (0.50) AURKAAURKBEGFRNTRK1
SCHEMBL3044547 0.77 SYK (0.33) AURKAAURKB
SCHEMBL26011193 0.74 SYK (0.42) AURKAAURKB
SCHEMBL26007684 0.74 PDE2A (0.33) AURKAAURKB
SCHEMBL26035235 0.74 SYK (0.32) AURKAAURKB
SCHEMBL3031923 0.72 IGF1R (0.45) AURKAAURKBEGFRNTRK1
SCHEMBL13220902 0.72 IGF1R (0.45) AURKAAURKBEGFRNTRK1
SCHEMBL26007557 0.71 SYK (0.40) AURKAAURKB
SCHEMBL26029263 0.71 SYK (0.42) AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154426-A1 CDK INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed