SCHEMBL26019255

SCHEMBL26019255

CS(=O)(=O)O[C@@H]1C[C@@H]2CN(OC(=O)c3ccccc3)C[C@@H]2C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
TSHR P16473 3/20 0.40
KMT2A Q03164 3/20 0.40
APOBEC3A P31941 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.38
FOLH1 Q04609 1/20 0.37
CYP2C9 P11712 1/20 0.36
MAPT P10636 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26019479 1.00 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL29346476 1.00 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL26019477 0.82 F2 (0.41) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL26018931 0.82 F2 (0.41) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL26317140 0.81 KMT2A (0.49) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL3728123 0.76 CARM1 (0.46) CHRNA7TSHRKMT2AAPOBEC3AAPOBEC3G
SCHEMBL25796422 0.75 F2 (0.47) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL25971778 0.75 CHRNA7 (0.41) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL29346477 0.74 GRIN1 (0.56) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL26019480 0.74 GRIN1 (0.52) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3974420-B1 N-ALKYLARYL-5-OXYHETEROARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B NOVARTIS AG (CH) 2023-08-16 EP disclosed